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How we can establish or improve Structure activity relationship(SAR) for the development of H1-Antihistamine drug?
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Solved in 2 steps
- Briefly discuss how we can improve pharmacodynamic properties of H1-Antihistamine drugs?How we can improve these parameters(isomerism, isosteric replacement) for the development of H1-Antihistamine drugs?What are the potential implications of genetic variations in drug-metabolizing enzymes on individual response and therapeutic outcomes in clinical pharmacology?
- What are the different methods for developing modified release drug delivery system ? Discuss about the matrix and encapsulation drug release systems. Please explain at your own words.How we can improve pharmacokinetic parameters for the development of H1-Antihistamine ? DiscussHow we can improve pharmacodynamic properties of H1-Antihistamine drugs?
- What properties of drug are relevant for developing modified release drug delivery formulation. Please briefly explain this at your own words.Please Write the Drug Discovery Process of Diltiazem? Please write at your own words.What are Targeted drug delivery systems ? Please explain the ideal properties of Targeted drug delivery systems?